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CAS:912444-00-9|ABT 888
- 产品货号:E-2024057817
- 发布时间:2024-06-03
- 产品CAS :912444-00-9
- 产品规格:mg(更多包装需求请咨询客服)
- 产品纯度:95%+
- 产品货期:现货下单后48小时内发货,定制产品4-8周。
- 运输条件:顺丰常规运输
产品详情
货号:E-2024057817
CAS:912444-00-9
规格:mg(更多包装需求请咨询客服)
纯度:95%+
生产商:试剂家
试剂家(www.empireagents.com) - 瑞禧生物旗下试剂品牌。致力于为全球客户提供高性价比的助力药物递送的产品服务。公司的奋斗目标是搭建一个国际知名的药物递送修饰平台,携手高端人才和所有合作伙伴,共同为人类各行各业的事业发展做出贡献!
Catalogue Number:A112580
Chemical Name:ABT 888
Synonyms:2-[(2R)-2-Methyl-2-pyrrolidinyl]-1H-benzimidazole-7-carboxamide; A 861695;
CAS Number:912444-00-9
Molecular Formula:C₁₃H₁₆N₄O
Appearance:Off-White to Dark Yellow Solid
Melting Point:>173°C (dec.)
Molecular Weight:244.29
Storage:4°C
Solubility:Methanol (Slightly), THF (Slightly)
Category:Research Tools; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
Applications:ABT-888 is a potent, orally bioavailable PARP-1/-2 inhibitor shown to potentiate DNA damaging agents. The ability to potentiate temozolomide (TMZ) and develop a biological marker for PARP inhibition was evaluated in vivo. Potent PARP inhibitor.
References:Virag, L., et al.: Pharmacol. Rev., 54, 375试剂家(www.empireagents.com)从未停止过技术的拓展与创新。凭借这充满进取的创新精神,我们已经为国内外高校、科研单位、材料研究中心、生物技术制药开发公司等等定制合成了各种功能化试剂,赢得了合作单位的长期信赖。
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