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CAS:1794960-29-4|rac-AS-703026-d5

  • 产品货号:E-2024063534
  • 发布时间:2024-06-13
  • 产品CAS :1794960-29-4
  • 产品规格:mg(更多包装需求请咨询客服)
  • 产品纯度:95%+
  • 产品货期:现货下单后48小时内发货,定制产品4-8周。
  • 运输条件:顺丰常规运输
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货号:E-2024063534
CAS:1794960-29-4
规格:mg(更多包装需求请咨询客服)
纯度:95%+
生产商:试剂家

试剂家(www.empireagents.com) - 瑞禧生物旗下试剂品牌。致力于为全球客户提供高性价比的助力药物递送的产品服务。公司的奋斗目标是搭建一个国际知名的药物递送修饰平台,携手高端人才和所有合作伙伴,共同为人类各行各业的事业发展做出贡献!
Catalogue Number:A780102
Chemical Name:rac-AS-703026-d5
Synonyms:N-[(2R,S)-2,3-Dihydroxypropyl-d5]-3-[(2-fluoro-4-iodophenyl)amino]-4-pyridinecarboxamide;
CAS Number:1794960-29-4
Alternate CAS #
1236699-92-5-unlabelled
Molecular Formula:C₁₅H₁₀D₅FIN₃O₃
Molecular Weight:436.23
Category:Standards; Isotopic Labeled Analogues; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
Applications:Labelled AS703026 (A780100). AS703026 is a novel, selective, orally bioavailable MEK1/2 inhibitor, in human multiple myeloma (MM). AS703026 induces pleiotropic anti-myeloma activity in vitro and in vivo. MEK inhibitors are useful in the treatment of hyperproliferative diseases, such as cancer, restenosis and inflammation.
References:Billadeau, D., et al.: Cancer Res., 55, 3640 (1995), Kolch, W., et al.: Biochem. J., 351, 289 (2000), Smith, M., et al.: Leukemia, 17, 274 (2003), Adjei, A., et al.: J. Clin. Oncol., 26, 2139 (2008),
试剂家(www.empireagents.com)从未停止过技术的拓展与创新。凭借这充满进取的创新精神,我们已经为国内外高校、科研单位、材料研究中心、生物技术制药开发公司等等定制合成了各种功能化试剂,赢得了合作单位的长期信赖。
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